Tyrosine kinase inhibitorFDA-approvedFirst-line

Brafiib

Generic name: dabrafenib

How it works

Blocks the BRAF V600E mutation in cancer cells, preventing uncontrolled cell growth.

Cancer types

MelanomaBRAF V600E-positive

Efficacy

In clinical trials, dabrafenib improved response rates in patients with BRAF V600E-positive melanoma, with a response rate of approximately 58%.

Side effects

Moderate

Side effects can be significant and may require dose adjustments or supportive medication, but the treatment is usually continued.

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.