CDK4/6 inhibitorFDA-approvedFirst-line

Ribociclib

How it works

Blocks the CDK4/6 enzymes, which are involved in cell growth and division.

Cancer types

Breast CancerHormone receptor-positive

Efficacy

Ribociclib has been shown to improve progression-free survival in patients with hormone receptor-positive metastatic breast cancer.

Side effects

Moderate

Side effects can be significant and may require dose adjustments or supportive medication, but the treatment is usually continued.

Evidence from research

StudyCancer typeStageEfficacy
Studying Ribociclib and Chemotherapy for High-Risk Breast CancerBreast Cancerphase-2Source →
Testing a Combination Treatment for HER2 Positive Breast CancerBreast Cancerphase-1Source →
Comparing a New Therapy to Chemotherapy for Early Breast CancerBreast Cancerphase-3Source →
Evaluating Leucogen to Prevent Low White Blood Cell Count in Breast Cancer Patients Taking RibociclibBreast Cancerphase-2Source →
Evaluating a New Treatment Combination for Advanced Breast CancerBreast Cancerphase-2Source →
Ribociclib and Hormone Therapy in Breast CancerBreast Cancerphase-3Source →
Assessing the Effectiveness and Safety of Ribociclib in Breast Cancer TreatmentBreast CancerpreclinicalSource →
Evaluating Patient Outcomes with Ribociclib in Early-Stage Breast CancerBreast CancerpreclinicalSource →
Study of Ribociclib and Hormone Therapy in Early Breast CancerBreast Cancerphase-3Source →
Testing Letrozole and Ribociclib in Early Breast CancerBreast Cancerphase-2Source →
Cyclin Dependent Kinase Inhibitors in Metastatic Breast CancerBreast CancerobservationalIn patients receiving palbociclib, a better median progression-free survival (PFS) was observed in patients with Eastern Cooperative Oncology Group (ECOG) performance status (PS) 1 (27.3 months,p-value <0.0001), de novo disease (17.5 months,p-value 0.0155), first line hormonal therapy (22.5 months,p-value <0.0001) and no prior chemotherapy (20.3 months,p-value 0.0001).Source →
Ribociclib and Letrozole Effective in Older Women with Advanced Breast CancerBreast CancerpreclinicalThe median progression-free survival was 36 months, and the breast cancer-specific survival rate at 24 and 36 months was 82% and 75%, respectively.Source →
Combining Ferulic Acid with Breast Cancer Drugs May Improve TreatmentBreast Cancerlab-studySource →
New Nanoparticle Delivery System for Breast Cancer TreatmentBreast Cancerlab-studyThe RIB-LNC exhibited a 1.31-fold and 3.09-fold reduction in IC values in MDA-MB-231 and MCF-7 cells, respectively, as compared to free RIB.Source →
New Treatment Combination Approved for High-Risk Breast CancerBreast Cancerphase-3The invasive disease-free survival at 36 months was 90.7% for Ribo + AI versus 87.6% for AI, with a hazard ratio of 0.75.Source →
CDK4/6 Inhibitors Linked to Cardiotoxic Events in Breast Cancer PatientsBreast CancerobservationalSource →
Ribociclib Improves Survival in Early Breast CancerBreast Cancerphase-3At 3 years, invasive disease-free survival was 90.4% with ribociclib plus an NSAI and 87.1% with an NSAI alone.Source →
CDK4/6 Inhibitors and Endocrine Therapy for Metastatic Breast CancerBreast Cancerphase-3Ribociclib combined with letrozole significantly improved PFS over letrozole alone.Source →
Targeted Liposomes Deliver Cancer Drug to Breast Cancer CellsBreast Cancerlab-studySource →
Comparing Two Cancer Treatments in Younger WomenBreast CancerobservationalThe median progression-free survival was 24.05 months for palbociclib and 24.41 months for ribociclib.Source →

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.