Hormone therapyFDA-approvedFirst-line

Tamoxifen

How it works

Blocks estrogen receptors on cancer cells, preventing growth signals and inhibiting cell division.

Cancer types

Breast CancerHormone receptor-positive

Efficacy

Clinical trials have demonstrated that tamoxifen can improve response rates and progression-free survival in patients with hormone receptor-positive breast cancer.

Side effects

Mild

Most people tolerate this treatment well. Side effects are generally manageable and do not require stopping treatment.

Evidence from research

StudyCancer typeStageEfficacy
Tamoxifen and Other Hormone Treatments for Invasive Breast CancerBreast Cancerphase-3Source →
Tamoxifen vs Z-Endoxifen in Advanced Breast CancerBreast Cancerphase-2Source →
Tamoxifen and Omega-3 for Breast Cancer RiskBreast Cancerphase-2Source →
Tamoxifen Dose Trial for Breast CancerBreast Cancerphase-2Source →
Breast Cancer Prevention TrialBreast Cancerphase-2Source →
Tamoxifen Side Effects Linked to Genetic Variants in South African Breast Cancer PatientsBreast CancerobservationalSource →
Tamoxifen-loaded Nanoparticles Improve Breast Cancer TreatmentBreast Cancerlab-studyThe particles were 6.21-fold more cytotoxic than free tamoxifen.Source →
Tamoxifen Drug Interactions Depend on Genetic Variation and Inhibitor StrengthBreast CancerobservationalSource →
Vaginal Tamoxifen May Help Postmenopausal Women with Vaginal Atrophy SymptomsBreast Cancerphase-2Women on vaginal tamoxifen were more likely to report no or minor symptoms after three months, OR 21.76 (95% CI 7.36 - 64.3).Source →
Tamoxifen Resistance in Breast Cancer: A Key Player IdentifiedBreast Cancerlab-studySource →
Tamoxifen and Endometrial Health in Breast Cancer PatientsBreast CancerobservationalSource →
Tamoxifen Linked to Uterine Cancer through Non-Genetic DriverOvarian Cancerlab-studySource →
Tamoxifen Resistance Overcome with New Cancer Treatment ApproachBreast Cancerlab-studySource →
Tamoxifen Resistance in Breast Cancer: New Insights into Metabolic ChangesBreast Cancerlab-studyDemethylation restored ASS1 expression and correspondingly reduced tamoxifen IC toward parental levels.Source →
New Nanoparticles Help Target Breast Cancer CellsBreast Cancerlab-studyBA@mPEGA FA BSA NPs reduced LCC9 cell IC by 2.29-fold (pH 6.5) versus free BA+TAM.Source →
Genetic Variants Affect Tamoxifen Use in Young Breast Cancer PatientsBreast CancerobservationalSource →
USP30's Role in Breast Cancer Progression and Resistance to TamoxifenBreast Cancerlab-studySource →
Hormone Therapy Side Effects in Breast Cancer PatientsBreast CancerobservationalSource →
Zeylonone May Help Overcome Tamoxifen Resistance in Breast CancerBreast Cancerlab-studySource →

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.