Hormone therapyFDA-approvedAdjuvant

Tamoxifen

How it works

Blocks estrogen receptors on cancer cells, preventing growth signals.

Cancer types

Breast CancerHormone receptor-positive

Efficacy

Tamoxifen has been shown to reduce the risk of breast cancer recurrence in hormone receptor-positive patients.

Side effects

Mild

Most people tolerate this treatment well. Side effects are generally manageable and do not require stopping treatment.

Evidence from research

StudyCancer typeStageEfficacy
miR-548as-5p May Help Overcome Tamoxifen Resistance in Breast CancerBreast Cancerlab-studySource →
Ovarian Function Suppression Reduces Breast Cancer Recurrence in Young WomenBreast Cancermeta-analysisSource →
Tamoxifen Hybrids Show Promise in Treating Triple-Negative Breast CancerBreast Cancerlab-studyCu-tamoxifen showed a more profound tumor-reducing potential than tamoxifen alone.Source →
Alternative Therapies and Breast Cancer Treatment AdherenceBreast CancerpreclinicalSource →
Combining Plant Extract and Tamoxifen May Help Reduce Cancer EnzymeBreast Canceranimal-studyThe combination of tamoxifen and E. bulbosa ethanol extract significantly reduced COX-2 levels to 3.86 ng/mL, close to the value observed in the negative control group (3.07 ng/mL).Source →
Low-Dose Tamoxifen May Help Prevent Breast CancerBreast Cancermeta-analysisThe overall mortality rate reduced after taking low-dose tamoxifen (p = 0.002).Source →
Tamoxifen and Other Hormone Treatments for Invasive Breast CancerBreast Cancerphase-3Source →
Tamoxifen vs Z-Endoxifen in Advanced Breast CancerBreast Cancerphase-2Source →
Tamoxifen Dose Trial for Breast CancerBreast Cancerphase-2Source →
Tamoxifen and Omega-3 for Breast Cancer RiskBreast Cancerphase-2Source →
Breast Cancer Prevention TrialBreast Cancerphase-2Source →
Tamoxifen Side Effects Linked to Genetic Variants in South African Breast Cancer PatientsBreast CancerobservationalSource →
Tamoxifen-loaded Nanoparticles Improve Breast Cancer TreatmentBreast Cancerlab-studyThe particles were 6.21-fold more cytotoxic than free tamoxifen.Source →
Tamoxifen Drug Interactions Depend on Genetic Variation and Inhibitor StrengthBreast CancerobservationalSource →
Vaginal Tamoxifen May Help Postmenopausal Women with Vaginal Atrophy SymptomsBreast Cancerphase-2Women on vaginal tamoxifen were more likely to report no or minor symptoms after three months, OR 21.76 (95% CI 7.36 - 64.3).Source →
Tamoxifen Resistance in Breast Cancer: A Key Player IdentifiedBreast Cancerlab-studySource →
Tamoxifen and Endometrial Health in Breast Cancer PatientsBreast CancerobservationalSource →
Rare Breast Cancer Recurrence After 46 Years of RemissionBreast CancerobservationalSource →
Tamoxifen Linked to Uterine Cancer through Non-Genetic DriverOvarian Cancerlab-studySource →
Tamoxifen Resistance Overcome with New Cancer Treatment ApproachBreast Cancerlab-studySource →
Tamoxifen Resistance in Breast Cancer: New Insights into Metabolic ChangesBreast Cancerlab-studyDemethylation restored ASS1 expression and correspondingly reduced tamoxifen IC toward parental levels.Source →
New Nanoparticles Help Target Breast Cancer CellsBreast Cancerlab-studyBA@mPEGA FA BSA NPs reduced LCC9 cell IC by 2.29-fold (pH 6.5) versus free BA+TAM.Source →
Genetic Variants Affect Tamoxifen Use in Young Breast Cancer PatientsBreast CancerobservationalSource →
Tamoxifen Therapy Benefits Vary by Menopausal Status in Breast CancerBreast Cancerphase-3In premenopausal patients, a statistically significant tamoxifen benefit was observed for lymph node-negative (adjusted hazard ratio [HR] = 0.46, 95% confidence interval [CI] = 0.24 to 0.87), progesterone receptor-positive (adjusted HR = 0.61, 95% CI = 0.41 to 0.91), and genomic low-risk tumors (adjusted HR = 0.47, 95% CI = 0.26 to 0.85) but only lasted beyond 10 years for genomic low-risk tumors.Source →
USP30's Role in Breast Cancer Progression and Resistance to TamoxifenBreast Cancerlab-studySource →
CYP2D6 Genes Linked to Breast Cancer OutcomesBreast Cancermeta-analysisSource →
Hormone Therapy Side Effects in Breast Cancer PatientsBreast CancerobservationalSource →
Antidepressant Use Changes After Breast Cancer TreatmentBreast CancerobservationalSource →
FoxO3a May Help Overcome Tamoxifen Resistance in Breast CancerBreast Cancerlab-studySource →
Rare Ovarian Cancer Treated with Tamoxifen for 10 YearsOvarian CancerobservationalSource →
Cost-Effectiveness of Breast Cancer Treatment in ChinaBreast Cancerphase-3Source →
Zeylonone May Help Overcome Tamoxifen Resistance in Breast CancerBreast Cancerlab-studySource →

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.