ChemotherapyFDA-approvedSecond-line

Trifluridine/tipiracil

How it works

Trifluridine is converted into FUTA in the body, which interferes with DNA replication and cell division, ultimately killing cancer cells.

Cancer types

Colorectal CancerAll patients

Efficacy

Studies show that trifluridine/tipiracil can improve overall survival in patients with metastatic colorectal cancer who have failed prior therapies.

Side effects

Moderate

Side effects can be significant and may require dose adjustments or supportive medication, but the treatment is usually continued.

Evidence from research

StudyCancer typeStageEfficacy
New Treatment Combination Shows Promise for Metastatic Colorectal CancerColorectal Cancerphase-2The objective response rate was 18.3%, and the disease control rate was 83.3%.Source →
Trifluridine/Tipiracil Treatment in Metastatic Colorectal CancerColorectal CancerobservationalMedian overall survival was 7.59 months.Source →
Trifluridine/Tipiracil Combinations Show Promise in Advanced Colorectal CancerColorectal CancerreviewMedian overall survival ranged 8.6-14.4 months and median progression-free survival 3.7-6.8 months with FTD/TPI plus bevacizumab in refractory mCRC.Source →

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.