Tyrosine kinase inhibitorPhase 3 trialInvestigational

Zanubrutinib

How it works

Blocks the Bruton's tyrosine kinase (BTK) protein, which is involved in the growth and survival of leukemia cells.

Cancer types

LeukemiaAll patients

Side effects

Moderate

Side effects can be significant and may require dose adjustments or supportive medication, but the treatment is usually continued.

Evidence from research

StudyCancer typeStageEfficacy
Testing Zanubrutinib and Rituximab for Chronic Lymphocytic Leukemia or Small Lymphocytic LymphomaLeukemiaphase-2Source →
Zanubrutinib Shows Promise in Rare Blood CancerLeukemiaobservationalSource →
Zanubrutinib and Sonrotoclax Combination for Rare Lymphoma in Underrepresented GroupsLeukemiaphase-1Source →
Investigating a New Treatment Combination for Untreated Chronic Lymphocytic LeukemiaLeukemiaphase-2Source →
New Treatment Combination for Untreated Chronic Lymphocytic LeukemiaLeukemiaphase-3Source →
Zanubrutinib, Obinutuzumab, and Venetoclax for CLL or SLLLeukemiaphase-2Source →
Study of CLL Treatment CombinationLeukemiaphase-3Source →
Comparing Zanubrutinib and Acalabrutinib in Relapsed CLLLeukemiaphase-3One progression was avoided per 10 patients treated (NNT=10) and one death per 15 patients treated (NNT=15) with zanubrutinib.Source →
New Study Compares Effectiveness of CLL TreatmentsLeukemiameta-analysisZanubrutinib had a significantly reduced risk of progression or death compared with ibrutinib (hazard ratio [HR], 0.49; 95% credible interval [CrI], 0.31-0.78).Source →
Zanubrutinib vs Ibrutinib for Chronic Lymphocytic Leukemia: Cost ComparisonLeukemiaphase-3Treating 8 patients with zanubrutinib instead of ibrutinib prevented 1 progression or death.Source →
Rare Side Effect of Cancer Drug ZanubrutinibLeukemiaobservationalSource →
Expert Panel Discusses Zanubrutinib Use in Chronic Lymphocytic LeukemiaLeukemiareviewSource →
Comparing Zanubrutinib and Ibrutinib for Leukemia TreatmentLeukemiameta-analysisSource →

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.