PARP inhibitorPhase 3 trialInvestigational

Lynparza (Olaparib)

Generic name: olaparib

How it works

Blocks the action of an enzyme called PARP, which helps repair DNA damage in cancer cells, leading to cell death.

Cancer types

Ovarian CancerBRCA1/2-mutated

Efficacy

Lynparza has been shown to improve progression-free survival in BRCA1/2-mutated ovarian cancer patients, with approximately 8 months of median progression-free survival in clinical trials.

Side effects

Mild

Most people tolerate this treatment well. Side effects are generally manageable and do not require stopping treatment.

Evidence from research

StudyCancer typeStageEfficacy
Olaparib and Abiraterone Combination Therapy for Prostate CancerProstate Cancerphase-2The 1-year radiographic progression-free survival rate was 77.7% (95% CI: 63.4-95.3%).Source →
New Compound Disrupts Cancer Gene ExpressionColorectal Cancerlab-studySource →
Testing Combination Therapy for Advanced Solid TumorsLung Cancerphase-1Source →
Studying Olaparib in Metastatic Prostate CancerProstate CancerpreclinicalSource →
Olaparib Study for Patients Who Have Completed Previous Oncology TrialsBreast Cancerphase-3Source →
Testing Olaparib with Radium-223 in Advanced Prostate CancerProstate Cancerphase-1Source →
Testing Ceralasertib in Combination with Other Treatments for Various CancersProstate Cancerphase-2Source →
Cediranib and Olaparib Combination Therapy for Advanced Solid TumorsBreast Cancerphase-2Source →
Testing Cediranib and Olaparib in Ovarian and Breast CancerBreast Cancerphase-1Source →
Testing Cediranib and Olaparib in Recurrent Ovarian CancerOvarian Cancerphase-2Source →
Testing New Treatments for Women with Recurrent Ovarian CancerOvarian Cancerphase-3Source →
Testing a Combination of Two Drugs for Recurrent Ovarian CancerOvarian Cancerphase-2Source →
Testing FPI-2265 and Olaparib for Metastatic Prostate CancerProstate Cancerphase-2Source →
Testing Radiotherapy and Immunotherapy for Small Cell Lung CancerLung Cancerphase-1Source →
Evaluating Olaparib in Chinese Patients with Advanced Prostate CancerProstate CancerpreclinicalSource →
Testing Olaparib and Pembrolizumab for Advanced Uveal MelanomaMelanomaphase-2Source →
Testing Combination Therapy for Advanced Solid TumorsLung Cancerphase-1Source →
Combining two treatments for advanced prostate cancerProstate Cancerphase-2Median radiographic progression-free survival was 5.0 months, and median overall survival was 19.1 months.Source →
Testing Olaparib for Ovarian Cancer TreatmentOvarian Cancerphase-3Source →
Olaparib for Relapsed/Refractory Acute Myeloid Leukemia or Myelodysplastic SyndromeLeukemiaphase-2Source →
Researchers Identify New Target to Enhance Prostate Cancer TreatmentProstate Cancerlab-studySource →
Curcumin Analogue and Olaparib Combination Shows Promise in Ovarian CancerOvarian Cancerlab-studySource →
New Combination Therapy Shows Promise in Treating Triple-Negative Breast CancerBreast Cancerlab-studyThe combination of Olaparib and Exemestane was able to achieve enhanced tumor growth inhibition in a murine xenograft model, greater than either drug employed as a single agent.Source →
TTK protein linked to resistance in ovarian cancer treatmentOvarian Cancerlab-studySource →
Olaparib plus bevacizumab in older ovarian cancer patients: manageable safety and quality of lifeOvarian Cancerphase-3Two years after randomization, mean Global Health Status and cognitive functioning seemed better with olaparib than bevacizumab alone (adjusted mean difference: +4.47 points and +4.82 points, respectively).Source →
Combining Cancer Treatments May Help Prostate Cancer PatientsProstate Cancerlab-studySource →
Combining Cancer Drugs Boosts Immune Response in Resistant Breast CancerBreast Cancerlab-studySource →
New Options for Treating Advanced Breast CancerBreast CancerreviewSource →
DRG2 levels predict response to PARP inhibitors in prostate cancer cellsProstate Cancerlab-studySource →
Olaparib Monotherapy Shows Promise in Lung Cancer TreatmentLung Cancermeta-analysisOlaparib monotherapy increased progression-free survival (PFS) level [ES= 7.76; 95% CI= 0.16 to 1.36; P=0.208].Source →
Olaparib Therapy Side Effects in UAE PatientsBreast CancerobservationalSource →
Olaparib vs Nonplatinum Chemotherapy in Ovarian CancerOvarian Cancerphase-3Overall survival with olaparib was similar to chemotherapy (median 34.9 and 32.9 months, respectively).Source →
Combining drugs may improve ovarian cancer treatmentOvarian Cancerlab-studyThe combined treatment allows a substantial dose reduction of olaparib rendering a strong synergistic effect.Source →
Olaparib Maintenance Therapy Shows Promise in Ovarian CancerOvarian CancerobservationalThe 1-year progression-free survival rate was 75.2% (95% CI, 63.4 to 89.2), and the median PFS was 21.0 months (95% CI, 13.8 to 28.2).Source →
Combining Cancer Drugs May Improve Treatment for Advanced Ovarian CancerOvarian Cancerlab-studySource →
Rare Lung Disease Linked to Cancer TreatmentBreast CancerobservationalSource →
Olaparib and Abiraterone Combination Therapy for Prostate CancerProstate CancerreviewSource →
gBRCA Testing and Olaparib in Pancreatic CancerPancreatic CancerobservationalThe best responses to platinum-based chemotherapy included a complete response in one patient (12.5%) and a partial response in seven patients (87.5%).Source →
Combination Cediranib and Olaparib Shows Activity in Ovarian CancerOvarian Cancerphase-2In platinum-sensitive ovarian cancer, the overall response rate was 77.1% and median progression-free survival was 16.4 months.Source →
Olaparib Maintenance Therapy in Ovarian Cancer: Biomarker AnalysisOvarian Cancerphase-3HRD-positive patients displayed greater median PFS [17.9 months (95% CI: 14.5-22.1)] than HRD-negative patients [9.2 months (95% CI: 7.5-13.8)].Source →
Olaparib Maintenance Therapy for Ovarian Cancer: A Study at Kurume University HospitalOvarian CancerobservationalThe median progression-free survival was 8.9 months, and the median overall survival was 27.1 months.Source →
Pancreatic Cancer Treatment Shows Promise in Rare Genetic CaseOvarian CancerobservationalSource →
CRABP2 May Reduce Effectiveness of Cancer Treatment OlaparibOvarian Cancerlab-studySource →
Inhibiting FSP1 Enhances Olaparib Sensitivity in Ovarian CancerOvarian Cancerlab-studySource →
Combining Olaparib and CDK12-IN-3 to Treat Ovarian CancerOvarian Cancerlab-studySource →
Researchers Identify Possible Cause of Cancer Treatment ResistancePancreatic Cancerlab-studySource →
New Treatment Combination for Advanced Prostate CancerProstate Cancerphase-3The median radiographic progression-free survival was 25 months for olaparib plus abiraterone versus 17 months for placebo plus abiraterone.Source →
Combining drugs may help overcome resistance to ovarian cancer treatmentOvarian Cancerlab-studySource →
Measuring PARP Inhibitors in Ovarian Cancer PatientsOvarian Cancerlab-studySource →
Choosing the Right Maintenance Therapy for Advanced Ovarian CancerOvarian Cancerphase-3Source →

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.