PARP inhibitorFDA-approvedSecond-line

Niraparib

How it works

Blocks the enzyme that helps repair damaged DNA, making it harder for cancer cells to grow and divide.

Cancer types

Pancreatic CancerBRCA-mutated
Ovarian CancerBRCA1/2-mutated

Efficacy

Niraparib has been shown to improve progression-free survival in BRCA1/2-mutated ovarian cancer patients, with a median progression-free survival of approximately 21 months.

Side effects

Mild

Most people tolerate this treatment well. Side effects are generally manageable and do not require stopping treatment.

Evidence from research

StudyCancer typeStageEfficacy
Testing Niraparib and Neratinib in Advanced Solid Tumors and Ovarian CancerOvarian Cancerphase-1Source →
Risk Factors for Niraparib-induced Anemia in Japanese Ovarian Cancer PatientsOvarian CancerobservationalSource →
Evaluating Niraparib for Ovarian Cancer TreatmentOvarian CancerpreclinicalSource →
Testing Niraparib in Ovarian Cancer Patients with Limited SpreadOvarian Cancerphase-2Source →
Heated Chemotherapy and Niraparib for Advanced Ovarian and Peritoneal CancersOvarian Cancerphase-3Source →
New Treatment Combination Shows Promise for Men with Advanced Prostate CancerProstate Cancerphase-3Median radiographic progression-free survival was 38.6 months in the niraparib + AAP group versus 8.3 months in the placebo + AAP group.Source →
Evaluating a New Treatment Combination for Recurrent Ovarian CancerOvarian Cancerphase-2Source →
Combination Therapy for Advanced Prostate CancerProstate Cancerphase-3Source →
Testing Niraparib and Copanlisib in Advanced Ovarian and Endometrial CancerOvarian Cancerphase-1Source →
Niraparib's Safety and Effectiveness in Ovarian Cancer TreatmentOvarian CancerobservationalSource →
Niraparib May Offer Better Progression-Free Survival for Ovarian Cancer PatientsOvarian CancerobservationalThe median progression-free survival was 13.77 months in the bevacizumab group.Source →
Niraparib May Lower Platelet Count in Ovarian Cancer PatientsOvarian CancerobservationalSource →
Niraparib Safety and Effectiveness in Older Patients with Tubo-Ovarian CancerOvarian CancerobservationalProgression-free survival was 12 months (95%CI: 2.0-25.0) for patients aged 50-64, 29 months (95%CI: 11.0-52.0) for patients aged 65-74, and 16 months (95%CI: 1.0-31.0) for patients aged 75 and older.Source →
Combining Medications May Help Prostate Cancer PatientsProstate Cancerphase-3The primary endpoint was met, with a significant improvement in radiographic progression-free survival observed, with a hazard ratio of 0.63.Source →
Ovarian Cancer Cells May Become More Sensitive to TreatmentOvarian Cancerlab-studyThe resistance indices for A2780/NRP and OVCAR3/NRP were 8.95 and 4.42, respectively.Source →
Corneal Deposits Linked to Cancer TreatmentOvarian CancerobservationalSource →
New Treatment Combination Shows Modest Progression-Free Survival Benefit in Advanced Ovarian CancerOvarian Cancerphase-3The primary endpoint was investigator-assessed progression-free survival (PFS) as per RECIST v1.1, with a median of 20.6 months in arm 3 versus 19.2 months in arm 2.Source →
Ovarian Cancer Treatment Linked to Heart Problems in Some PatientsOvarian Cancerlab-studySource →
Niraparib Shows Promise in Treating Advanced MelanomaMelanomaphase-2The disease control rate was 64%.Source →
Rare Blood Platelet Deficiency Linked to Cancer DrugOvarian CancerobservationalSource →
Real-world study of ovarian cancer treatment reveals patient experiencesOvarian CancerobservationalSource →
Combining Cancer Drugs May Improve Ovarian Cancer TreatmentOvarian Cancerphase-3Patients receiving maintenance niraparib who reported concomitant use of statins exhibited significantly improved PFS compared with those on placebo with concomitant statins (HR = 0.34; P < 0.001; median PFS 18.2 vs. 6.0 months).Source →
Individualized Dose of Niraparib Reduces Hematologic Adverse Event CostsOvarian Cancerphase-3The total mean calculated AE management cost per patient was $12,987.71 with the FSD and $6744.93 with the ISD.Source →
Real-world outcomes of ovarian cancer patients on niraparib-bevacizumab maintenance therapyOvarian Cancerphase-2Median time to treatment discontinuation was 11.8 months (95% CI 8.7 to 13.5), and median time to next treatment was 14.1 months (95% CI 11.3 to 16.6).Source →
Niraparib Side Effects: Researchers Identify Risk Factors for Nausea and VomitingOvarian CancerobservationalSource →
Niraparib Maintenance Therapy in Ovarian Cancer: Long-Term Survival ResultsOvarian Cancerphase-3The 5-year PFS rate numerically favored niraparib in the overall (niraparib, 22%; placebo, 12%) and HRd populations (niraparib, 35%; placebo, 16%).Source →
Niraparib May Improve Survival in Ovarian Cancer PatientsOvarian CancerobservationalMedian overall survival was 24.1 months in the niraparib group and 18.4 months in the active surveillance group.Source →
Niraparib Efficacy and Safety in Japanese Women with Ovarian CancerOvarian Cancerphase-2Confirmed objective response rate was 60.0% (90% confidence interval [CI]=39.4-78.3)Source →
Combining Cancer Treatments May Improve EffectivenessOvarian Cancerlab-studySource →
PARP Inhibitors Linked to Cardiovascular Risks in Ovarian Cancer PatientsOvarian CancerobservationalSource →
Adjusting Dose of Cancer Drug Niraparib May Improve SafetyOvarian Cancerphase-3Source →
Niraparib as Maintenance Therapy for Ovarian Cancer in JapanOvarian CancerobservationalSource →
Niraparib Dose Adjusted for Safety in Ovarian Cancer PatientsOvarian Cancerphase-3Source →
Niraparib Efficacy and Safety in Ovarian CancerOvarian CancerobservationalMedian overall survival was 30 months, and median progression-free survival was 8 months.Source →
New Treatment Combination Shows Modest Activity in Advanced Ovarian CancerOvarian Cancerphase-2The objective response rate was 17.1% (80% CI, 9.8 to 27.0), including one complete response (2.4%).Source →
Rare Lung Disease Linked to Ovarian Cancer DrugOvarian CancerobservationalSource →
Niraparib Tested for Rare Genetic Mutation in Gastrointestinal CancersPancreatic Cancerphase-2Source →
Niraparib therapy linked to increased creatinine levels in ovarian cancer patientsOvarian CancerobservationalSource →
Measuring PARP Inhibitors in Ovarian Cancer PatientsOvarian Cancerlab-studySource →
Choosing the Right Maintenance Therapy for Advanced Ovarian CancerOvarian Cancerphase-3Source →

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.