Tyrosine kinase inhibitorFDA-approvedSecond-line

Palbociclib

How it works

Blocks the CDK4/6 enzymes that drive cell division in cancer cells, allowing the body's natural repair mechanisms to take over.

Cancer types

Breast CancerHormone receptor-positive

Efficacy

Studies have shown that palbociclib can improve progression-free survival and overall survival in patients with hormone receptor-positive breast cancer.

Side effects

Moderate

Side effects can be significant and may require dose adjustments or supportive medication, but the treatment is usually continued.

Evidence from research

StudyCancer typeStageEfficacy
Using Text Messages to Help People Take Palbociclib for Breast CancerBreast CancerpreclinicalSource →
Testing Palbociclib and Binimetinib in RAS-Mutant CancersPancreatic Cancerphase-2Source →
New Long-Acting Palbociclib Injection for Metastatic Breast CancerBreast Cancerlab-studySource →
Palbociclib in Metastatic Prostate Cancer: A Clinical TrialProstate Cancerphase-2Source →
Lab Test Models Breast Cancer Cells to Study Palbociclib EffectivenessBreast Cancerlab-studySource →
New Insights into Treating Low-Grade Ovarian CancerOvarian Cancerlab-studySource →
Palbociclib and Neutropenia in Metastatic Breast CancerBreast CancerobservationalThe 30-month PFS rate was 75% with the dose of 100 mg, 90.9% with 75 mg, and 97.2% with the dose of 125 mg.Source →
Palbociclib's Potential in Leukemia TreatmentLeukemiareviewSource →
Palbociclib Effectiveness in Indian Breast Cancer PatientsBreast CancerobservationalThe real-world response rate and the real-world clinical benefit rate across treatment lines were 68% and 75.3%, respectively.Source →
Intermittent Palbociclib Use in Metastatic Breast Cancer During Economic CrisisBreast CancerobservationalIntermittent discontinuation statistically reduces PFS by 26%.Source →
Real-world effectiveness of palbociclib in breast cancer treatmentBreast Cancermeta-analysisFirst-line palbociclib+AI MMPFS (22.5 months, 95% CI = 19.5 to 31.8) aligned with PALOMA-1/2 pooled mPFS (23.9, 95% CI = 20.2 to 27.6).Source →
Palbociclib and Endocrine Therapy for Metastatic Breast Cancer in JapanBreast CancerobservationalThe median progression-free survival was 26.6 months.Source →
Comparing Two Cancer Treatments in Younger WomenBreast CancerobservationalThe median progression-free survival was 24.05 months for palbociclib and 24.41 months for ribociclib.Source →

This information is provided for general education only and is not medical advice. Always consult a qualified healthcare professional before making treatment decisions.