Treatments

An overview of cancer treatments across types — from approved standard-of-care options to agents under active investigation. Select any treatment to learn how it works and which cancer types it applies to.

First-line

5-Fluorouracil

Chemotherapy

Moderate side effects

Adriamycin

Chemotherapy

Severe side effects

Adriamycin (Doxorubicin)

Chemotherapy

Severe side effects

Alecensa

Tyrosine kinase inhibitor

Moderate side effects

Alectinib

Tyrosine kinase inhibitor

Mild side effects

Alimta

Chemotherapy

Moderate side effects

Alimta (Pemetrexed)

Chemotherapy

Severe side effects

Apalutamide

Hormone therapy

Moderate side effects

Aromatase inhibitors (e.g. Anastrozole)

Hormone therapy

Mild side effects

Aromatase inhibitors (e.g. Letrozole)

Hormone therapy

Mild side effects

Avastin

Monoclonal antibody

Severe side effects

Azacitidine

Chemotherapy

Moderate side effects

Bicalutamide

Hormone therapy

Mild side effects

Brafi

Tyrosine kinase inhibitor

Severe side effects

Brafiib

Tyrosine kinase inhibitor

Moderate side effects

BRAF/MEK inhibitor combination

Tyrosine kinase inhibitor

Moderate side effects

BRAF/MEK Inhibitor Combination (Dabrafenib + Trametinib)

Tyrosine kinase inhibitor

Moderate side effects

BRAF/MEK Inhibitor Combination (Encorafenib + Binimetinib)

Tyrosine kinase inhibitor

Moderate side effects

BRAF V600E inhibitor (Encorafenib)

Tyrosine kinase inhibitor

Moderate side effects

Capecitabine

Chemotherapy

Moderate side effects

Carboplatin

Chemotherapy

Severe side effects

Carboplatin + Paclitaxel

Chemotherapy

Severe side effects

Cemiplimab

Monoclonal antibody

Moderate side effects

Cetuximab

Monoclonal antibody

Moderate side effects

Chemotherapy (e.g. Doxorubicin)

Chemotherapy

Severe side effects

Cisplatin

Chemotherapy

Severe side effects

Cotellic

Tyrosine kinase inhibitor

Moderate side effects

Crizotinib

Tyrosine kinase inhibitor

Moderate side effects

Cytarabine

Chemotherapy

Severe side effects

Dabrafenib

Tyrosine kinase inhibitor

Moderate side effects

Dacomitinib

Tyrosine kinase inhibitor

Severe side effects

Darolutamide

Hormone therapy

Mild side effects

Docetaxel

Chemotherapy

Severe side effects

Encorafenib

Tyrosine kinase inhibitor

Moderate side effects

Fludarabine

Chemotherapy

Severe side effects

FOLFIRINOX

Chemotherapy

Severe side effects

FOLFOX

Chemotherapy

Severe side effects

Gefitinib

Tyrosine kinase inhibitor

Moderate side effects

Gemcitabine

Chemotherapy

Moderate side effects

Gemcitabine + nab-paclitaxel

Chemotherapy

Moderate side effects

Gilotrif

Tyrosine kinase inhibitor

Moderate side effects

Idarubicin

Chemotherapy

Severe side effects

Imatinib

Tyrosine kinase inhibitor

Moderate side effects

Ipilimumab

Immunotherapy / CTLA-4 inhibitor

Severe side effects

Keytruda

Immunotherapy / PD-1 inhibitor

Mild side effects

L-asparaginase

Chemotherapy

Severe side effects

Leucovorin

Chemotherapy

Mild side effects

Leuprolide

Hormone therapy

Mild side effects

Lupron

Hormone therapy

Moderate side effects

Midostaurin

Tyrosine kinase inhibitor

Moderate side effects

Nab-paclitaxel

Chemotherapy

Moderate side effects

Osimertinib

Tyrosine kinase inhibitor

Moderate side effects

Paclitaxel

Chemotherapy

Severe side effects

Pemetrexed

Chemotherapy

Severe side effects

Pertuzumab

Monoclonal antibody

Mild side effects

Platinum-based chemotherapy

Chemotherapy

Severe side effects

Platinum-based chemotherapy (e.g., carboplatin, cisplatin)

Chemotherapy

Severe side effects

Relugolix

Hormone therapy

Mild side effects

Rituximab

Monoclonal antibody

Mild side effects

Ruxolitinib

JAK inhibitor

Moderate side effects

Squibb's Tarceva

Tyrosine kinase inhibitor

Moderate side effects

Tarceva

Tyrosine kinase inhibitor

Moderate side effects

Trastuzumab

Monoclonal antibody

Mild side effects

Vemurafenib

Tyrosine kinase inhibitor

Moderate side effects

Vincristine

Chemotherapy

Severe side effects

Vizimpro

Tyrosine kinase inhibitor

Severe side effects

Xalkori

Tyrosine kinase inhibitor

Moderate side effects

Xeloda

Chemotherapy

Moderate side effects

Yervoy

Monoclonal antibody

Severe side effects

Zelboraf

Tyrosine kinase inhibitor

Moderate side effects

Second-line

Abiraterone

Hormone therapy

Moderate side effects

Abiraterone acetate

Hormone therapy

Moderate side effects

Ado-trastuzumab emtansine

Monoclonal antibody-drug conjugate

Severe side effects

Alpelisib

PI3K inhibitor

Moderate side effects

Bevacizumab

Monoclonal antibody

Severe side effects

Binimetinib

Tyrosine kinase inhibitor

Moderate side effects

Blinatumomab

Monoclonal antibody

Moderate side effects

Bosutinib

Tyrosine kinase inhibitor

Moderate side effects

Braftovi

Tyrosine kinase inhibitor

Moderate side effects

Brentuximab vedotin

Monoclonal antibody-drug conjugate

Moderate side effects

Cabazitaxel

Chemotherapy

Severe side effects

Carfilzomib

Proteasome inhibitor

Severe side effects

Cladribine

Chemotherapy

Severe side effects

Clofarabine

Chemotherapy

Severe side effects

Cobimetinib

Tyrosine kinase inhibitor

Moderate side effects

Dasatinib

Tyrosine kinase inhibitor

Moderate side effects

Durvalumab

Immunotherapy / PD-1 inhibitor

Mild side effects

Enzalutamide

Hormone therapy

Moderate side effects

Erbitux

Monoclonal antibody

Severe side effects

Erlotinib

Tyrosine kinase inhibitor

Moderate side effects

Everolimus

mTOR inhibitor

Moderate side effects

FOLFIRI

Chemotherapy

Severe side effects

Fulvestrant

Hormone therapy

Moderate side effects

Imfinzi

Immunotherapy / PD-1 inhibitor

Mild side effects

Inotuzumab ozogamicin

Monoclonal antibody

Severe side effects

Iressa

Tyrosine kinase inhibitor

Mild side effects

Irinotecan

Chemotherapy

Moderate side effects

Jevtana

Chemotherapy

Severe side effects

Lonsurf

Chemotherapy

Severe side effects

Lorbrena

Tyrosine kinase inhibitor

Moderate side effects

Lorlatinib

Tyrosine kinase inhibitor

Moderate side effects

Lutetium-177 PSMA

Radiopharmaceutical therapy

Mild side effects

Lutetium-177 vipivotide tetraxetan

Radiopharmaceutical

Severe side effects

Lutetium Lu 177 vipivotide tetraxetan

Radiopharmaceutical

Severe side effects

Mekinist

Tyrosine kinase inhibitor

Moderate side effects

Mektovi

Tyrosine kinase inhibitor

Moderate side effects

MM-398

Chemotherapy

Moderate side effects

Neratinib

Tyrosine kinase inhibitor

Moderate side effects

Niraparib

PARP inhibitor

Mild side effects

Nivolumab

Immunotherapy / PD-1 inhibitor

Mild side effects

Nivolumab + Ipilimumab

Monoclonal antibody

Severe side effects

Nubeqa

Hormone therapy

Moderate side effects

Opdivo

Immunotherapy / PD-1 inhibitor

Mild side effects

Oxaliplatin

Chemotherapy

Severe side effects

Palbociclib

CDK4/6 inhibitor

Moderate side effects

Panitumumab

Monoclonal antibody

Moderate side effects

Pembrolizumab + Axitinib

Immunotherapy / Combination

Moderate side effects

Ponatinib

Tyrosine kinase inhibitor

Severe side effects

Radium-223

Radiopharmaceutical

Mild side effects

Radium-223 dichloride

Radiotherapy

Moderate side effects

Radium Ra 223 dichloride

Radiopharmaceutical

Severe side effects

Regorafenib

Tyrosine kinase inhibitor

Severe side effects

Ribociclib

CDK4/6 inhibitor

Moderate side effects

Rucaparib

PARP inhibitor

Mild side effects

S-1

Chemotherapy

Moderate side effects

Stivarga

Tyrosine kinase inhibitor

Severe side effects

Tafinlar + Mekinist

Tyrosine kinase inhibitor

Moderate side effects

Tagrisso

Tyrosine kinase inhibitor

Moderate side effects

Taxotere

Chemotherapy

Severe side effects

Tecentriq

Immunotherapy / PD-L1 inhibitor

Mild side effects

Topotecan

Chemotherapy

Moderate side effects

Trametinib

Tyrosine kinase inhibitor

Moderate side effects

Trastuzumab-DM1

Monoclonal antibody-drug conjugate

Moderate side effects

Trifluridine/tipiracil

Chemotherapy

Moderate side effects

Vectibix

Monoclonal antibody

Moderate side effects

Xtandi

Hormone therapy

Moderate side effects

Zaltrap

Monoclonal antibody

Severe side effects

Zanubrutinib

BTK inhibitor

Moderate side effects

Zykadia

Tyrosine kinase inhibitor

Moderate side effects

Zytiga

Hormone therapy

Severe side effects

Adjuvant

Investigational

Abemaciclib

CDK4/6 inhibitor

Moderate side effects

Apatinib

Tyrosine kinase inhibitor

Moderate side effects

APC-4037

Hormone therapy

Moderate side effects

ARV-110

Hormone therapy

Moderate side effects

Atezolizumab

Immunotherapy / PD-L1 inhibitor

Moderate side effects

Avelumab

Immunotherapy / PD-1 inhibitor

Mild side effects

Bempegaldesleukin

Immunotherapy / IL-2 agonist

Severe side effects

Cabozantinib

Tyrosine kinase inhibitor

Moderate side effects

Capivasertib

PARP inhibitor

Moderate side effects

Capmatinib

Tyrosine kinase inhibitor

Moderate side effects

Cediranib

Tyrosine kinase inhibitor

Severe side effects

Ceritinib

Tyrosine kinase inhibitor

Moderate side effects

Decitabine

Chemotherapy

Severe side effects

Dinutuximab

Monoclonal antibody

Moderate side effects

Dinutuximab beta

Monoclonal antibody

Mild side effects

Dostarlimab

Immunotherapy / PD-1 inhibitor

Moderate side effects

Doxorubicin

Chemotherapy

Severe side effects

Durvalumab/ezetimibe

Immunotherapy / PD-1 inhibitor + Cholesterol absorption inhibitor

Mild side effects

Durvalumab + tremelimumab

Immunotherapy

Mild side effects

Enasidenib

IDH2 inhibitor

Moderate side effects

Fedratinib

JAK2 inhibitor

Moderate side effects

Gilteritinib

FLT3 inhibitor

Moderate side effects

Ibrutinib

BTK inhibitor

Moderate side effects

Idecabtagene vicleucel

CAR-T cell therapy

Severe side effects

Isturisa

Hormone therapy

Moderate side effects

Ivosidenib

IDH1 inhibitor

Moderate side effects

Ketek

Chemotherapy

Severe side effects

Kisqali

CDK4/6 inhibitor

Moderate side effects

Ladiratuzumab vedotin

Monoclonal antibody-drug conjugate

Moderate side effects

Lapatinib

Tyrosine kinase inhibitor

Severe side effects

Larotrectinib

Tyrosine kinase inhibitor

Mild side effects

Liso-cel

CAR-T cell therapy

Severe side effects

Luspatercept

Erythropoiesis-stimulating agent

Mild side effects

Lynparza

PARP inhibitor

Mild side effects

Lynparza (Olaparib)

PARP inhibitor

Mild side effects

Margetuximab

Monoclonal antibody

Moderate side effects

MM-151

Monoclonal antibody

Mild side effects

Mobocertinib

Tyrosine kinase inhibitor

Moderate side effects

Nab-selinexor

Chemotherapy

Severe side effects

NBTXR3

Radiosensitizer

Mild side effects

Necitumumab

Monoclonal antibody

Moderate side effects

Olaparib

PARP inhibitor

Mild side effects

Olaratumab

Monoclonal antibody

Moderate side effects

PARP inhibitor

PARP inhibitor

Moderate side effects

Pazopanib

Tyrosine kinase inhibitor

Moderate side effects

PDR001

Immunotherapy / PD-1 inhibitor

Moderate side effects

Pembrolizumab

Immunotherapy / PD-1 inhibitor

Moderate side effects

Pembrolizumab + ipilimumab

Combination therapy

Severe side effects

Pembrolizumab + Lenvatinib

Monoclonal antibody + Tyrosine kinase inhibitor

Severe side effects

Pembrolizumab + Nivolumab

Immunotherapy / PD-1 inhibitor

Mild side effects

Pembrolizumab + Vemurafenib

Monoclonal antibody, Tyrosine kinase inhibitor

Severe side effects

Platinum-based chemotherapy (e.g. Carboplatin)

Chemotherapy

Severe side effects

Platinum-based chemotherapy (e.g., carboplatin, cisplatin, oxaliplatin)

Chemotherapy

Severe side effects

Pluvicto

Radiation therapy

Severe side effects

Pralsetinib

Tyrosine kinase inhibitor

Severe side effects

Ramucirumab

Monoclonal antibody

Moderate side effects

regorafenib + bevacizumab

Tyrosine kinase inhibitor + Monoclonal antibody

Severe side effects

Regorafenib ( investigational combination )

Tyrosine kinase inhibitor

Severe side effects

regorafenib + Lonsurf

Tyrosine kinase inhibitor + Chemotherapy

Severe side effects

Sacituzumab Govitecan

Monoclonal antibody

Severe side effects

Selpercatinib

Tyrosine kinase inhibitor

Moderate side effects

Selumetinib

MEK inhibitor

Moderate side effects

Sorafenib

Tyrosine kinase inhibitor

Moderate side effects

Sotorasib

Tyrosine kinase inhibitor

Moderate side effects

Tafasitamab

Monoclonal antibody

Moderate side effects

Talazoparib

PARP inhibitor

Mild side effects

TAS-120

PI3K inhibitor

Moderate side effects

Temozolomide

Chemotherapy

Moderate side effects

Tiragolumab

Immunotherapy / TIGIT inhibitor

Mild side effects

Tisagenlecleucel

CAR-T cell therapy

Severe side effects

Tislelizumab

Immunotherapy / PD-1 inhibitor

Mild side effects

Tisotumab Vedotin

Monoclonal antibody-drug conjugate

Severe side effects

Tucatinib

Tyrosine kinase inhibitor

Moderate side effects

Tumor Treating Fields (TTF) with Optune

Electromagnetic therapy

Mild side effects

Venetoclax

BCL-2 inhibitor

Severe side effects

Vosaroxin

Anthraquinone

Severe side effects

Zoliflodine

Immunotherapy / PD-1 inhibitor

Moderate side effects

Other

Treatment information is provided for general education only — not medical advice.